OALib Journal期刊
ISSN: 2333-9721
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Discovery and Optimization of Potent, Selective, and in Vivo Efficacious 2-Aryl Benzimidazole BCATm Inhibitors
DOI: 10.1021/acsmedchemlett.5b00389
Alain Daugan, Anne-Benedicte Boullay, Arthur Beljean, Christopher C. Arico-Muendel, Christopher Kollmann, Chun-Wa Chung, Clare Hobbs, Donald O. Somers, Edwige Nicodeme, Emily Blazensky, Eric Boursier, Eric Humphries, Flora Sundersingh, Hongfeng Deng, Jeffrey A. Messer, Jing Chai, Jingye Zhou, Kenny Herry, Myriam Ajakane, Nerina Dodic, Paul Carter, Ryan Bingham, Sarah
E. Smith, Svetlana
L. Belyanskaya, Van Loc Nguyen, Yun Ding
Keywords: BCATm, branched chain amino acids (BCAAs), DNA Encoded Library, ELT, 2-aryl benzimidazole
Abstract:
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