%0 Journal Article %T Discovery and Optimization of Potent, Selective, and in Vivo Efficacious 2-Aryl Benzimidazole BCATm Inhibitors %A Alain Daugan %A Anne-Benedicte Boullay %A Arthur Beljean %A Christopher C. Arico-Muendel %A Christopher Kollmann %A Chun-Wa Chung %A Clare Hobbs %A Donald O. Somers %A Edwige Nicodeme %A Emily Blazensky %A Eric Boursier %A Eric Humphries %A Flora Sundersingh %A Hongfeng Deng %A Jeffrey A. Messer %A Jing Chai %A Jingye Zhou %A Kenny Herry %A Myriam Ajakane %A Nerina Dodic %A Paul Carter %A Ryan Bingham %A Sarah E. Smith %A Svetlana L. Belyanskaya %A Van Loc Nguyen %A Yun Ding %J Archive of "ACS Medicinal Chemistry Letters". %D 2016 %R 10.1021/acsmedchemlett.5b00389 %K BCATm %K branched chain amino acids (BCAAs) %K DNA Encoded Library %K ELT %K 2-aryl benzimidazole %U https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4834658/