OALib Journal期刊
ISSN: 2333-9721
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GluN2A-Selective Pyridopyrimidinone Series of NMDAR
Positive Allosteric Modulators with an Improved in Vivo Profile
DOI: 10.1021/acsmedchemlett.6b00388
Aijun Lu, Benjamin D. Sellers, Bianca M. Liederer, Cuong Q. Ly, David H. Hackos, Elisia Villemure, Emile Plise, Gauri Deshmukh, Guosheng Wu, Heidi J. A. Wallweber, Jacob B. Schwarz, Jesse
E. Hanson, Kimberly Scearce-Levie, Matthew Volgraf, Mingcui Liu, Patrick
J. Lupardus, Po-wai Yuen, Shun Zhang, Suzanne Tay, Tzu-Ming Wang, Xifeng Luo, Yu Jiang
Keywords: NMDAR, PAM, AMPAR, allosteric, potentiator, selectivity, brain concentration, CNS, EPSP
Abstract:
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