OALib Journal期刊
ISSN: 2333-9721
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Discovery
of Pyrazolo[1,5-a]pyrimidine TTK Inhibitors:
CFI-402257 is a Potent, Selective, Bioavailable
Anticancer Agent
DOI: 10.1021/acsmedchemlett.5b00485
Dan Chi-Chia Lin, Donald E. Awrey, Grace Ng, Graham
C. Fletcher, Henry W. Pauls, Irina Beletskaya, Jacqueline M. Mason, Mark R. Bray, Miklos Feher, Narendra
Kumar Patel, Nickolay Y. Chirgadze, Olga Plotnikova, Peter B. Sampson, Radoslaw Laufer, Reza Kiarash, Richard Brokx, Richard Hodgson, Sze-Wan Li, Tak W. Mak, Wei Qiu, Xin Wei, Yi Che, Yong Liu, Yunhui Lang
Keywords: TTK inhibitors, CFI-402257, pyrazolo[1,5-a]pyrimidines, 11/2 type inhibitors
Abstract:
Full-Text
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