%0 Journal Article %T Discovery of Pyrazolo[1,5-a]pyrimidine TTK Inhibitors: CFI-402257 is a Potent, Selective, Bioavailable Anticancer Agent %A Dan Chi-Chia Lin %A Donald E. Awrey %A Grace Ng %A Graham C. Fletcher %A Henry W. Pauls %A Irina Beletskaya %A Jacqueline M. Mason %A Mark R. Bray %A Miklos Feher %A Narendra Kumar Patel %A Nickolay Y. Chirgadze %A Olga Plotnikova %A Peter B. Sampson %A Radoslaw Laufer %A Reza Kiarash %A Richard Brokx %A Richard Hodgson %A Sze-Wan Li %A Tak W. Mak %A Wei Qiu %A Xin Wei %A Yi Che %A Yong Liu %A Yunhui Lang %J Archive of "ACS Medicinal Chemistry Letters". %D 2016 %R 10.1021/acsmedchemlett.5b00485 %K TTK inhibitors %K CFI-402257 %K pyrazolo[1 %K 5-a]pyrimidines %K 11/2 type inhibitors %U https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4948001/