OALib Journal期刊
ISSN: 2333-9721
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Fragment-Based Discovery of a Selective and Cell-Active Benzodiazepinone
CBP/EP300 Bromodomain Inhibitor (CPI-637)
DOI: 10.1021/acsmedchemlett.6b00075
Alexander M. Taylor, Alexandre C?té, Andrea G. Cochran, Andrew
R. Conery, Brian K. Albrecht, Christopher G. Nasveschuk, Dong Yu, E. Megan Flynn, Eneida Pardo, F. Anthony Romero, Fen Yan, Gladys de Leon
Boenig, Hariharan Jayaram, Henry Lu, James
E. Audia, James R. Kiefer, Jeremy Murray, Jeremy Setser, Jian Wang, Jiangpeng Liao, Laura Zawadzke, Leslie A. Dakin, Maureen H. Beresini, Michael C. Hewitt, Nico Cantone, Oscar W. Huang, Patricia J. Keller, Richard Pastor, Richard T. Cummings, Robert J. Sims, III, Steve Bellon, Steven Magnuson, Susan Kaufman, Terry
D. Crawford, Tommy Lai, Vickie Tsui, Wenfeng Liu, Xiaoqin Zhu, Xiaoyu Zhu, Yingjie Li, Yongyun Wang, Yves Leblanc, Zhaowu Xu, Zhongguo Chen
Keywords: Bromodomain, CREBBP, CBP, EP300, benzodiazepinone
Abstract:
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