%0 Journal Article
%T Fragment-Based Discovery of a Selective and Cell-Active Benzodiazepinone
CBP/EP300 Bromodomain Inhibitor (CPI-637)
%A Alexander M. Taylor
%A Alexandre C£¿t¨¦
%A Andrea G. Cochran
%A Andrew
R. Conery
%A Brian K. Albrecht
%A Christopher G. Nasveschuk
%A Dong Yu
%A E. Megan Flynn
%A Eneida Pardo
%A F. Anthony Romero
%A Fen Yan
%A Gladys de Leon
Boenig
%A Hariharan Jayaram
%A Henry Lu
%A James
E. Audia
%A James R. Kiefer
%A Jeremy Murray
%A Jeremy Setser
%A Jian Wang
%A Jiangpeng Liao
%A Laura Zawadzke
%A Leslie A. Dakin
%A Maureen H. Beresini
%A Michael C. Hewitt
%A Nico Cantone
%A Oscar W. Huang
%A Patricia J. Keller
%A Richard Pastor
%A Richard T. Cummings
%A Robert J. Sims
%A III
%A Steve Bellon
%A Steven Magnuson
%A Susan Kaufman
%A Terry
D. Crawford
%A Tommy Lai
%A Vickie Tsui
%A Wenfeng Liu
%A Xiaoqin Zhu
%A Xiaoyu Zhu
%A Yingjie Li
%A Yongyun Wang
%A Yves Leblanc
%A Zhaowu Xu
%A Zhongguo Chen
%J Archive of "ACS Medicinal Chemistry Letters".
%D 2016
%R 10.1021/acsmedchemlett.6b00075
%K Bromodomain
%K CREBBP
%K CBP
%K EP300
%K benzodiazepinone
%U https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4867486/