OALib Journal期刊
ISSN: 2333-9721
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Discovery and Optimization of Macrocyclic Quinoxaline-pyrrolo-dihydropiperidinones
as Potent Pim-1/2 Kinase Inhibitors
DOI: 10.1021/acsmedchemlett.5b00403
Andrew S. Tasker, Anthony B. Reed, Bethany
K. Mattson, Bin Wu, Bradley Herberich, Brian A. Lanman, Christine E. Sastri, Christopher Mohr, Dean Hickman, Frank Chavez, Jr., Hui-Ling Wang, J. Russell Lipford, Jeffrey T. Winston, Jie Chen, Jimmy Laszlo, III, Karen Rex, Kristin L. Andrews, Liping H. Pettus, Matthew R. Lee, Nadia Guerrero, Paul Wang, Qiong Wu, Ryan P. Wurz, Tian Wu, Victor J. Cee, Yang Xu, Yen Nguyen, Yihong Zhou
Keywords: Pim kinase inhibitor, multiple myeloma, KMS-12-BM, macrocycle
Abstract:
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