%0 Journal Article %T Discovery and Optimization of Macrocyclic Quinoxaline-pyrrolo-dihydropiperidinones as Potent Pim-1/2 Kinase Inhibitors %A Andrew S. Tasker %A Anthony B. Reed %A Bethany K. Mattson %A Bin Wu %A Bradley Herberich %A Brian A. Lanman %A Christine E. Sastri %A Christopher Mohr %A Dean Hickman %A Frank Chavez %A Jr. %A Hui-Ling Wang %A J. Russell Lipford %A Jeffrey T. Winston %A Jie Chen %A Jimmy Laszlo %A III %A Karen Rex %A Kristin L. Andrews %A Liping H. Pettus %A Matthew R. Lee %A Nadia Guerrero %A Paul Wang %A Qiong Wu %A Ryan P. Wurz %A Tian Wu %A Victor J. Cee %A Yang Xu %A Yen Nguyen %A Yihong Zhou %J Archive of "ACS Medicinal Chemistry Letters". %D 2016 %R 10.1021/acsmedchemlett.5b00403 %K Pim kinase inhibitor %K multiple myeloma %K KMS-12-BM %K macrocycle %U https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4834646/