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甾体与萜类的结构修饰以及三嗪类药物稳定性研究
The Structural Modification of Steroids and Terpenes and the Stability of Triazines

DOI: 10.12677/HJCET.2021.114029, PP. 214-218

Keywords: 甾体类,结构修饰,药理活性,稳定性
Steroids
, Structural Modification, Pharmacological Activity, Stability

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Abstract:

甾体与萜类以及三嗪类药物一般都具有比较复杂的结构,为增大其利用率,从而可以对其进行结构改造,来利用其产物的药理活性进行研究。以此类的活性化合物为母体,再对其结构修饰,从而能获得具有更高活性以及低毒性的化合物。另一方面,对三嗪类药地克珠利口服液进行处方筛选并制备,再对其进行相关稳定性试验,以便探讨此药物制剂的稳定性与评价。
Steroids, terpenes, and triazine drugs generally have relatively complex structures. In order to increase their utilization, they can be structurally modified to use the pharmacological activities of their products for research. Using this type of active compound as a parent and then modifying its structure, a compound with higher activity and low toxicity can be obtained. On the other hand, make the prescription screening and preparation of the triazine drug diclazuril oral liquid, and then related stability tests on it, in order to explore the stability and evaluation of the drug formulation.

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