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OALib Journal期刊
ISSN: 2333-9721
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-  2016 

Pharmacological characterization of a novel potent, selective, and orally active phosphodiesterase 10A inhibitor, PDM‐042 [(E)‐4‐(2‐(2‐(5,8‐dimethyl‐[1,2,4]triazolo[1,5‐a]pyrazin‐2‐yl)vinyl)‐6‐(pyrrolidin‐1‐yl)pyrimidin‐4‐yl)morpholine] in rats: potential for the treatment of schizophrenia

DOI: 10.1002/prp2.241

Keywords: Antipsychotics, catalepsy, occupancy, PDE10A, PDM‐042, schizophrenia

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