OALib Journal期刊
ISSN: 2333-9721
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2,8-Disubstituted-1,6-Naphthyridines and 4,6-Disubstituted-Isoquinolines with
Potent, Selective Affinity for CDK8/19
DOI: 10.1021/acsmedchemlett.6b00022
Christian Rink, Christina Esdar, Daniel Schwarz, Dirk Wienke, Djordje Musil, Felix Rohdich, Florence I. Raynaud, Jimmy Sejberg, Julian Blagg, Kai Schiemann, Klaus Urbahns, Mark A. Honey, Mark Stubbs, Michael Busch, Oliver Poeschke, Paul A. Clarke, Paul Czodrowski, Paul Workman, Richard Schneider, Rosemary Burke, Suzanne A. Eccles
Keywords: CDK8, CDK19, mediator complex, kinase inhibitor, aldehyde oxidase
Abstract:
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