Development of a Potent, Specific CDK8 Kinase Inhibitor
Which Phenocopies CDK8/19 Knockout Cells
DOI: 10.1021/acsmedchemlett.5b00278
Elisabeth
V. Schneider,
Elizabeth
M. Blackwood,
James R. Kiefer,
Jiansheng Wu,
Kevin R. Clark,
Klaus Maskos,
Krista Bowman,
Laurent Salphati,
Linda Orren,
Mark L. McCleland,
Maureen H. Beresini,
Michael F. T. Koehler,
Philippe Bergeron,
Ron Firestein,
Steve Schmidt
Keywords: CDK8, cyclin C, kinase inhibitor
Abstract:
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