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药学学报 2010
hiventryinhibitors:progressindevelopmentandapplication, PP. 131-140 Abstract: thisreviewdiscussesrecentprogressinthedevelopmentofanti-hivagents,withemphasisonsmallmoleculehiv-1entryinhibitors.？theentryinhibitorsprimarilytargethiv-1envelopeglycoproteinsorthecellularreceptors,cd4andchemokinereceptors.？twooftheentryinhibitors,enfuvirtideandmaraviroc,havebeenapprovedbytheusfdaforaidstherapy.？thedrugresistanceassociatedwithsomeoftheentryinhibitorswillalsobediscussed.
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