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化学进展  1999 

新型镇痛剂地棘蛙素的化学和药理

Keywords: 地棘蛙素,全合成,类似物,非阿片类镇痛剂,构效关系

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Abstract:

本文评述了新型非阿片类强效镇痛剂地棘蛙素的化学和药理研究的进展。从地棘蛙素全合成研究、类似物制备、药理学行为和构效关系等几方面介绍了国际上研究的热点,并对今后的研究动向进行了讨论。

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