Surade S, Blundell T L. Chem. Biol., 2012, 19 (1): 42.
[2]
Craik D J, Fairlie D P, Liras S, Price D. Chem. Biol. Drug Des., 2013, 81 (1): 136.
[3]
Danho W, Swistok J, Khan W, Chu X J, Cheung A, Fry D, Sun H, Kurylko G, Rumennik L, Cefalu J, Cefalu G, Nunn P. Adv. Exp. Med. Biol., 2009, 611: 467.
[4]
Vlieghe P, Lisowski V, Martinez J, Khrestchatisky M. Drug Discov. Today, 2010, 15 (1/2): 40.
[5]
Hamman J H, Enslin G M, Kotzé A F. BioDrugs, 2005, 19 (3): 165.
[6]
Góngora-Benítez M, Tulla-Puche J, Albericio F. Chem. Rev., 2014, 114 (2): 901.
[7]
Pattabiraman V R, Bode J W. Nature, 2011, 480: 471.
[8]
Kent S B H. Chem. Soc. Rev., 2009, 38: 338.
[9]
Cui H K, Guo Y, He Y, Wang F L, Chang H N, Wang Y J, Wu F M, Tian C L, Liu L. Angew. Chem. Int. Ed., 2013, 52: 9558.
[10]
Zheng J S, Chang H N, Shi J, Liu L. Sci. China Chem., 2012, 55: 64.
[11]
Petcher T J, Weber H, Rüegger A. Helv. Chim. Acta, 1976, 59 (5): 1480.
[12]
Loosli H R, Kessler H, Oschkinat H, Weber H P, Petcher T J, Widmer A. Helv. Chim. Acta, 1985, 68: 682.
[13]
Kessler H, Loosli H R, Oschkinat H. Helv. Chim. Acta, 1985, 68: 661.
[14]
Kessler H, Gehrke M, Lautz J, K?ck M, Seebach D, Thaler A. Biochem. Pharmacol., 1990, 40 (1): 169.
[15]
Saska I, Gillon A D, Hatsugai N, Dietzgen R G, Hara-Nishimura I, Anderson M A, Craik D J. J. Biol. Chem., 2007, 282 (40): 29721.
[16]
Zheng J S, Tang S, Guo Y, Chang H N, Liu L. ChemBioChem, 2012, 13 (4): 542.
[17]
Conlan B F, Gillon A D, Craik D J, Anderson M A. Biopolymers, 2010, 94 (5): 573.
[18]
Saether O, Craik D J, Campbell I D, Sletten K, Juul J, Norman D G. Biochemistry, 1995, 34 (13): 4147.
[19]
Henriques S T, Huang Y H, Rosengren K J, Franquelim H G, Carvalho F A, Johnson A, Sonza S, Tachedjian G, Castanho M A, Daly N L, Craik D J. J. Biol. Chem., 2011, 286 (52): 24231.
[20]
Dechantsreiter M A, Planker E, Math? B, Lohof E, H?lzemann G, Jonczyk A, Goodman S L, Kessler H. J. Med. Chem., 1999, 42 (16): 3033.
[21]
Doedens L, Opperer F, Cai M, Beck J G, Dedek M, Palmer E, Hruby V J, Kessler H. J. Am. Chem. Soc., 2010, 132 (23): 8115.
[22]
Yan L M, Tatarek-Nossol M, Velkova A, Kazantzis A, Kapurniotu A. Proc. Natl. Acad. Sci. U. S. A., 2006, 103 (7): 2046.
[23]
Biron E, Chatterjee J, Ovadia O, Langenegger D, Brueggen J, Hoyer D, Schmid H A, Jelinek R, Gilon C, Hoffman A, Kessler H. Angew. Chem. Int. Ed., 2008, 47 (14): 2595.
Moellering R E, Cornejo M, Davis T N, Del Bianco C, Aster J C, Blacklow S C, Kung A L, Gilliland D G, Verdine G L, Bradner J E. Nature, 2009, 462 (7270): 182.
[27]
Cui H K, Zhao B, Li Y H, Guo Y, Hu H, Liu L, Chen Y G. Cell Res., 2013, 23: 581
[28]
高帅(Gao S), 郭叶(Guo Y), 李海燕(Li H Y), 方葛敏(Fang G M). 化学进展(Prog. Chem.), 2014, 26 (1): 100.
[29]
Fawell S, Seery J, Daikh Y, Moore C, Chen L L, Pepinsky B, Barsoum J. Proc. Natl. Acad. Sci. U.S.A., 1994, 91(2): 664.
[30]
Zheng J S, Tang S, Huang Y C, Liu L. Acc. Chem. Res., 2013, 46 (11): 2475.
[31]
Wang P, Dong S, Shieh J H, Peguero E, Hendrickson R, Moore M A S, Danishefsky S J. Science, 2013, 342: 1357.
[32]
Zheng J S, Tang S, Qi Y K, Wang Z P, Liu L. Nat. Protoc., 2013, 8 (12): 2483.
[33]
Fang G M, Li Y M, Shen F, Huang Y C, Li J B, Lin Y, Cui H K, Liu L. Angew. Chem. Int. Ed., 2011, 50 (33): 7645.
[34]
Huang Y C, Li Y M, Chen Y, Pan M, Li Y T, Yu L, Guo Q X, Liu L. Angew. Chem. Int. Ed., 2013, 52: 4858.
[35]
Zheng J S, Chang H N, Wang F L, Liu L. J. Am. Chem. Soc., 2011, 133 (29): 11080.
[36]
Fang G M, Wang J X, Liu L. Angew. Chem. Int. Ed., 2012, 51: 10347.
[37]
Shao Y, Lu W, Kent S B H. Tetrahedron Lett., 1998, 39: 3911.
[38]
Chen J, Warren J D, Wu B, Chen G, Wan Q, Danishefsky S J. Tetrahedron Lett., 2006, 47: 1969.
Dittmann J, Wenger R M, Kleinkauf H, Lawen A. J. Biol. Chem., 1994, 269 (4): 2841.
[41]
Handschumacher R E, Harding M W, Rice J, Drugge R J, Speicher D W. Science, 1984, 226 (4674): 544.
[42]
Vine W, Bowers L D. CRC Crit. Rev. Clin. Lab. Sci., 1987, 25: 275.
[43]
el Tayar N, Mark A E, Vallat P, Brunne R M, Testa B, van Gunsteren W F. J. Med. Chem., 1993, 36 (24): 3757.
[44]
Wong C T, Rowlands D K, Wong C H, Lo T W, Nguyen G K, Li H Y, Tam J P. Angew. Chem. Int. Ed., 2012, 51 (23): 5620.
[45]
Greenwood K P, Daly N L, Brown D L, Stow J L, Craik D J. Int. J. Biochem. Cell Biol., 2007, 39 (12): 2252.
[46]
Contreras J, Elnagar A Y, Hamm-Alvarez S F, Camarero J A. J. Control. Release, 2011, 155 (2): 134.
[47]
Cascales L, Henriques S T, Kerr M C, Huang Y H, Sweet M J, Daly N L, Craik D J. J. Biol. Chem., 2011, 286 (42): 36932.
[48]
Knipp G T, Vander Velde D G, Siahaan T J, Borchardt R T. Pharm. Res., 1997, 14 (10): 1332.
[49]
Gudmundsson O S, Jois S D, Vander Velde D G, Siahaan T J, Wang B, Borchardt R T. J. Pept. Res., 1999, 53 (4): 383.
[50]
Boguslavsky V, Hruby V J, O'Brien D F, Misicka A, Lipkowski A W. J. Pept. Res., 2003, 61 (6): 287.
[51]
Rezai T, Yu B, Millhauser G L, Jacobson M P, Lokey R S. J. Am. Chem. Soc., 2006, 128 (8): 2510.
[52]
Rezai T, Bock J E, Zhou M V, Kalyanaraman C, Lokey R S, Jacobson M P. J. Am. Chem. Soc., 2006, 128 (43): 14073.
[53]
White T R, Renzelman C M, Rand A C, Rezai T, McEwen C M, Gelev V M, Turner R A, Linington R G, Leung S S, Kalgutkar A S, Bauman J N, Zhang Y, Liras S, Price D A, Mathiowetz A M, Jacobson M P, Lokey R S. Nat. Chem. Biol., 2011, 7 (11): 810.
[54]
Beck J G, Chatterjee J, Laufer B, Kiran M U, Frank A O, Neubauer S, Ovadia O, Greenberg S, Gilon C, Hoffman A, Kessler H. J. Am. Chem. Soc., 2012, 134 (29): 12125.
[55]
Gunasekera S, Foley F M, Clark R J, Sando L, Fabri L J, Craik D J, Daly N L. J. Med. Chem., 2008, 51 (24): 7697.
[56]
Ji Y, Majumder S, Millard M, Borra R, Bi T, Elnagar A Y, Neamati N, Shekhtman A, Camarero J A. J. Am. Chem. Soc., 2013, 135 (31): 11623.
[57]
Schafmeister C E, Po J, Verdine G L. J. Am. Chem. Soc., 2000, 122 (24): 5891.
[58]
Walensky L D, Kung A L, Escher I, Malia T J, Barbuto S, Wright R D, Wagner G, Verdine G L, Korsmeyer S J. Science, 2004, 305 (5689): 1466.
[59]
Danial N N, Walensky L D, Zhang C Y, Choi C S, Fisher J K, Molina A J, Datta S R, Pitter K L, Bird G H, Wikstrom J D, Deeney J T, Robertson K, Morash J, Kulkarni A, Neschen S, Kim S, Greenberg M E, Corkey B E, Shirihai O S, Shulman G I, Lowell B B, Korsmeyer S J. Nat. Med., 2008, 14 (2): 144.
[60]
Muppidi A, Doi K, Edwardraja S, Drake E J, Gulick A M, Wang H G, Lin Q. J. Am. Chem. Soc., 2012, 134 (36): 14734
[61]
Derossi D, Joliot A H, Chassaing G, Prochiantz A. J. Biol. Chem., 269 (14): 10444.
[62]
Morris M C, Depollier J, Mery J, Heitz F, Divita G. Nat. Biotechnol., 2001, 19 (12): 1173.
[63]
Mitchell D J, Kim D T, Steinman L, Fathman C G, Rothbard J B. J. Pept. Res., 56 (5): 318.
[64]
Richard J P, Melikov K, Vives E, Ramos C, Verbeure B, Gait M J, Chernomordik L V, Lebleu B. J. Biol. Chem., 2003, 278 (1): 585.
[65]
Ter-Avetisyan G, Tünnemann G, Nowak D, Nitschke M, Herrmann A, Drab M, Cardoso M C. J. Biol. Chem., 2009, 284 (6): 3370.
[66]
Tünnemann G, Ter-Avetisyan G, Martin R M, St?ckl M, Herrmann A, Cardoso M C. J. Pept. Sci., 2008, 14 (4): 469.
[67]
Liu T, Liu Y, Kao H Y, Pei D. J. Med. Chem., 2010, 53 (6): 2494.
[68]
Kanovsky M, Raffo A, Drew L, Rosal R, Do T, Friedman F K, Rubinstein P, Visser J, Robinson R, Brandt-Rauf P W, Michl J, Fine R L, Pincus M R. Proc. Natl. Acad. Sci. U.S.A., 2001, 98 (22): 12438.
[69]
Do T N, Rosal R V, Drew L, Raffo A J, Michl J, Pincus M R, Friedman F K, Petrylak D P, Cassai N, Szmulewicz J, Sidhu G, Fine R L, Brandt-Rauf P W. Oncogene, 2003, 22 (10): 1431.
[70]
Li C, Pazgier M, Liu M, Lu W Y, Lu W. Angew. Chem. Int. Ed., 2009, 48 (46): 8712.
[71]
L?ttig-Tünnemann G, Prinz M, Hoffmann D, Behlke J, Palm-Apergi C, Morano I, Herce H D, Cardoso M C. Nat. Commun., 2011, 2: 453.
[72]
Mandal D, Nasrolahi Shirazi A, Parang K. Angew. Chem. Int. Ed., 2011, 50 (41): 9633.
[73]
Nasrolahi Shirazi A, Tiwari R, Chhikara B S, Mandal D, Parang K. Mol. Pharm., 2013, 10 (2): 488.
[74]
Nasrolahi Shirazi A, Tiwari R K, Oh D, Banerjee A, Yadav A, Parang K. Mol. Pharm., 2013, 10 (5): 2008.
[75]
Qian Z, Liu T, Liu Y Y, Briesewitz R, Barrios A M, Jhiang S M, Pei D. ACS Chem. Biol., 2013, 8 (2): 423.
[76]
Chan D I, Prenner E J, Vogel H J. Biochim. Biophys. Acta, 2006, 1758 (9): 1184.
[77]
Rothbard J B, Jessop T C, Lewis R S, Murray B A, Wender P A. J. Am. Chem. Soc., 2004, 126 (31): 9506.
[78]
Rothbard J B, Kreider E, VanDeusen C L, Wright L, Wylie B L, Wender P A. J. Med. Chem., 2002, 45 (17): 3612.