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化学进展  1999 

核蛋白的生物功能及核肽的合成和应用

Keywords: 核蛋白,核肽,生物学效应,复制,合成,抗肿瘤药物,抗病毒药物

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Abstract:

核蛋白或核肽是一类其侧链羟基通过磷酸二酯键连接到DNA或RNA的3′或5′端的天然生物大分子,具有广泛的生物学效应,包括DNA及RNA的复制、DNA的转录、插入、缺失和重组等。核肽也指合成的核蛋白结合位点的片断,作为一种新的工具既可用于研究核蛋白产生生物效应的机理,又为开发新一类抗病毒、抗肿瘤药物开辟了道路。

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