OALib Journal期刊
ISSN: 2333-9721
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实体瘤中的低氧区与低氧选择性药物研究进展
Keywords: 肿瘤,低氧,低氧选择性,钴(III)络合物,氮芥
Abstract:
降低抗肿瘤药物的毒性是开发新药的重中之重.本文介绍一种设计抗癌新药的新思路即低氧选择性药物.对肿瘤中低氧区产生的原因,对放疗和化疗的影响,以及克服它的方法作了阐述,着重对低氧选择性药物的研究进展作了评述,并指出该药物的发展前景.
References
[1] | [ 1 ] Moulder J E , Rockwell S. Int . J . Radiat . Oncol . Biol . Phys ,1984 , 10 : 695 —712
|
[2] | [ 2 ] Achintya K S , Dhiren R. Adv. Prug Delivery Rew. , 1996 , 19 :241 —273
|
[3] | [ 3 ] Dische S. Radiotherap. Oncol . , 1985 , 3 : 97 —115
|
[4] | [ 4 ] Graeber T G, Osinanjao C , Jacks T, et al . Nature , 1996 , 379(6560) :88 —91
|
[5] | [ 6 ] 杨频(Yang P) , 高飞(Gao F) . 生物无机化学原理,第1 版.北京: 科学出版社,2002. 561 —563
|
[6] | [ 8 ] 艾春玲(Ai C L) . 实用肿瘤学杂志(Journal of Practical Oncology) , 2002 ,26 : 160
|
[7] | Twentyman P R. Cancer Treat . Rep. , 1976 , 60 : 1719 —1722
|
[8] | Barranco S C , Novak J K. Cancer Res. , 1974 , 34 : 1616 —1618
|
[9] | Barranco S C , Navak J K, Humphrey R M. Cancer Res. , 1973 ,33 : 691 —694
|
[10] | 高远红( Gao Y H) . 国外医学肿瘤学分册( Foreign Medical Sciences , Cancer Section) ,1999 , 26 : 270 —273
|
[11] | Jeremic B , Djueic L , Mijatovic L. Cancer , 1991 , 68 : 21 —38
|
[12] | Rockwell S , Irvin C G, Kelly M et al . Int . J . Radiat . Oncol .Biol . Phys. , 1992 , 22 : 87 —93
|
[13] | 朱广迎(Zhu G Y) , 张邻康( Zhang L K) . 徐州医学院学报(Journal of Xuzhou Medical College) , 1994 , 14 : 92
|
[14] | Sartorelli A C. Biochem. Pharmacol . , 1986 , 35 : 67 —69
|
[15] | Denny W A , Wilson W R. Cancer Metastasis Rev. , 1993 , 12 :135 —151
|
[16] | Sinhababu A K, Thakker D R. Advanced Drugs Delivery Review ,1996 , 19 : 241 —273
|
[17] | Tannock I F , Rotin D. Cancer Res. 1989 , 49 : 4373 —4384
|
[18] | Lewis D F V. Xenobiotica , 1989 , 19 : 341 —356
|
[19] | Ware D C , Siim B G, Robinson K G, Denny W A , Brothers P L ,Clark G R. Inorg. Chem. , 1991 , 30 : 3750 —3757
|
[20] | Ware D C , Palmer D B , Wilson W R , Denny W A. J . Med.Chem. , 1993 , 36 : 1839 —1846
|
[21] | Ware D C , Brothers P J , Clark G R , Denny W A , Palmer B D ,Wilson W R. J . Chem. Soc. , Dalton Trans. , 2000 , 925 —932
|
[22] | Ware D C , Palmer H R , Brothers P F , Rickard C E F , Wilson W R , Denny WA. J . Inorg. Biochem. , 1997 , 215 —224
|
[23] | Blower P J , Dilworth J R , Maurer R I , Mullen GD , Reynolds C A , Zheng Y F. J . Inorg. Biochem. , 2001 , 85 : 15 —22
|
[24] | 阎军(Yang J ) ,崔海萍(Cui H P) ,杨频(Yang P) ,化学研究与应用(Chemical Research and Application) ,2003 , 15 : 71 —74
|
[25] | [ 5 ] Zhong H , Agani F , Baccala A A , et al . Cancer Res. , 1998 ,58 : 5280 —5284
|
[26] | [ 7 ] 郭瑞中(Guo R Z) . 重庆医学(Chongqing Medical) ,2002 , 31 :428
|
[27] | [ 9 ] Hockel M, Schlenger K, Mitze M, et al . Semin in Radiat Oncol . , 1996 , 6 : 3 —9
|
[28] | Ciaccia A J . Semin in Radiat Oncol . , 1996 , 6 : 46 —58
|
[29] | Teicher B A , Lazo J S , Sartorelli A C. Cancer Res. , 1981 , 41 :73 —81
|
[30] | Teicher B A , Holden S A , Rose C M. J . Natl . Cancer Inst . ,1985 , 75 : 1129 —1133
|
[31] | Keyes S R , Rockwell S , Sartorelli A C. Cancer Res. , 1985 , 45 :3645 —3654
|
[32] | Oya N , Shibamoto Y, Sesni K, et al . Int . J . Radiat . Oncol .Biol . Phys. , 1995 , 33 : 119 —127
|
[33] | 解荷芝( Xie H Z) . 药学进展( Progress in Pharmaceutical Science) , 1997 ,21 (2) : 83 —88
|
[34] | Lin A J , Cosby A , Shansky C W, Sartorelli A C. J . Med.Chem. , 1972 , 15 : 1247 —1252
|
[35] | Lin A J , Pardini R S , Coaby L A , Lillis B , Shansky C W,Sartorelli A C. J . Med. Chem. , 1973 , 16 : 1268 —1271
|
[36] | Kennedy K A , Teicher B A , Rockwell S , Sartorelli A C. Biochem Parmacol . , 1980 , 29 : 1 —8
|
[37] | 李德华(Li D H) . 浙江肿瘤( Zhejiang Oncology) , 1999 , 5 :134 —135
|
[38] | William A , Denny W A , Wilson W R. Cancer and Metastasis Reviews , 1993 , 12 : 135 —151
|
[39] | 阎军( Yang J ) . 山西大学硕士论文(Master Dissertations of Shanxi University) . 1997
|
[40] | Chaplin D J , Acker M D , Olive P L. Int . J . Radiat . Oncol .Biol . Phys. , 1989 , 16 : 1131 —1135
|
[41] | Palmer B D , Wilson W R , Pullen S M, Denny W A. J . Med.Chem. , 1990 , 33 : 112 —121
|
[42] | Brophy G T, Sladek N E. Biochem. Pharmacol . , 1983 , 32 :79 —84
|
[43] | Skarsgard L D , Chaplin D J , Wilson D J , Skwarchuk M W,Vinczan A , Kristl J . Int . J . Radiat . Oncol . Biol . Phys. , 1992 ,22 : 737 —741
|
[44] | Tannock I. Cancer Treat Rep. , 1978 , 62 : 1117 —1133
|
[45] | Wilman D E V , Connors A T. Molecular Aspects of Anticancer Drug Action (eds. Neidle S , Waring MJ ) . London : McMillan ,1983. 1 —34
|
[46] | 赵广华(Zhao G H) . 山西大学硕士论文(Master Dissertations of Shanxi University) . 1995
|
[47] | Hendry P , Ludi A. Adv. Inorg. Chem. , 1990 , 35 : 117 —198
|
[48] | Keyes S R , Reimbrook D C , Fracasso P M, Rockwell S , Sligar S G, Sartorelli A C. Adv. Enzyme Reg. , 1985 , 23 : 291 —307
|
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