Johnson S M, Wiseman R L, Sekijima Y, Green N S, Adamski-Werner S L, Kelly J W. Acc. Chem. Res., 2005, 38: 911.
[2]
Haupt H, Heide K. Experientia, 1966, 22: 449.
[3]
Palaninathan S K. Curr. Med. Chem., 2012: 2324.
[4]
Blake C C, Geisow M J, Oatley S J, Rerat B, Rerat C. J. Mol. Bio., 1978, 121: 339.
[5]
Lei M, Yang M F, Huo S H. J. Struct. Biol., 2004, 148: 153.
[6]
Wojtczak A, Cody V, Luft J R, Pangborn W. Acta Crystallogr D, 1996, 52: 758.
[7]
Nencetti S, Orlandini E. Curr. Med. Chem., 2012, 19: 2356.
[8]
Hurshman A R, White J T, Powers E T, Kelly J W. Biochem., 2004, 43: 7365.
[9]
Liu K, Cho H S, Lashuel H A, Kelly J W, Wemmer D E. Nat. Struct. Bio., 2000, 7: 4.
[10]
Lauro A, Diago Usò T, Masetti M, Di Benedetto F, Cautero N, De Ruvo N, Dazzi A, Quintini C, Begliomini B, Siniscalchi A, Ramacciato G, Risaliti A, Miller C M, Pinna A D. Transpl. Proc., 2005, 37: 2214.
[11]
Hornsten R, Wiklund U, Olofsson B O, Hensen S M, Suhr O B. Transplantation, 2004, 78: 112.
[12]
Ando Y, Ueda M. Curr. Med. Chem., 2012, 19: 2312
[13]
Zhao L J, Zhang L R, Lei M. Sci. China-Chem., 2013, 56: 1550.
[14]
Baures P W, Peterson S A, Kelly J W. Bioorg. Med. Chem., 1998, 6(8): 1389.
[15]
Razavi H, Palaninathan S K, Powers E T, Wiseman R L, Purkey H E, Mohamedmohaideen N N, Deechongkit S, Chiang K P, Dendle M T A, Sacchettini J C, Kelly J W. Angew. Chem. Int. Edit., 2003, 42(24): 2758.
[16]
Johnson S M, Petrassi H M, Palaninathan S K, Mohamedmohaideen N N, Purkey H E, Nichols C, Chiang K P, Walkup T, Sacchettini J C, Sharpless K B, Kelly J W. J. Med. Chem., 2005, 48(5): 1576.
[17]
Armen R S, Alonso D O V, Daggett V. Structure, 2004, 12: 1847.
[18]
Armen R S, Demarco M L, Alonso D O V, Daggett V. Proc. Natl. Acad. Sci. U. S. A., 2004, 101: 11622.
[19]
Pauling L, Corey R B. Proc. Natl. Acad. Sci. U. S. A., 1951, 37(5): 251.
[20]
Yang M F, Lei M, Bruschweiler R, Huo S H. Biophy. J, 2005, 89: 433.
[21]
Yang M F, Yordanov B, Levy Y, Bruschweiler R, Huo S H. Biochem., 2006, 45: 11992.
[22]
Hammarstrom P, Schneider F, Kelly J W. Science, 2001, 293(5539): 2459.
[23]
Lim K H, Dyson H J, Kelly J W, Wright P E. J. Mol. Bio., 2013, 425(6): 977.
[24]
徐筱杰(Xu X J), 侯廷军(Hou T J), 乔学斌(Qiao X B), 章威(Zhang W). 计算机辅助药物分子设计(Computer-Aided Drug Design). 北京: 化学工业出版社(Beijing: Chemical Industry Press), 2004. 325.
[25]
Maia F, Almeida M R, Gales L, Kijjoa A, Pinto M M M, Saraiva M J, Damas A M. Biochem. Pharmaco., 2005, 70: 1861.
[26]
Gupta S, Chhibbe M, Sinha S, Surolia A. J. Med. Chem., 2007, 50: 5589.
[27]
Rossi M, Caruso F, Opazo C, Salciccioli J. J. Agric. Food. Chem., 2008, 56: 10557.
[28]
Connelly S, Choi S, Johnson S M, Kelly J W, Wilson I A. Cur. Opin. Struc. Bio., 2010, 20: 54.
[29]
Palaninathan S K, Mohamedmohaideen N N, Orlandini E, Ortore G, Nencetti S, Lapucci A, Rossello A, Freundlich J S, Sacchettini J C. PLoS One, 2009, 4: e6290.
[30]
Cao J, Lin Y, Guo L H, Zhang A Q, Wei Y, Yang Y. Toxicology, 2010, 277: 20.
[31]
Zhu L L, Xu X J. Chinese J. Chem., 2003, 21(3): 261.
[32]
Jana M W, Patrik L A, Marja H L, Pim E G L, Stefan P J L, Timo H. Toxicological Sci., 2009, 109: 206.
[33]
Blasi D, Arsequell G, Valencia G, Nieto J, Planas A, Pinto M, Centeno N B, Abad Z C, Quintana J. Mol. Inform., 2011, 30: 161.
[34]
Natesan S, Wang T S, Lukacova V, Bartus V, Khandelwal A, Balaz S. J. Chem. Inf. Model, 2011: 1132.
[35]
Pinto M, Blasi D, Nieto J, Arsequell G, Valencia G, Planas A, Centeno N B, Quintana J, Centeno N B. Amyloid, 2011, 18: 51.
[36]
Choi S, Ong D S T, Kelly J W. J. Am. Chem. Soc., 2010, 132: 1359.
[37]
Johnson S M, Connelly S, Fearns C, Powers E T, Kelly J W. J. Mol. Bio., 2012, 421: 185.
[38]
Hamilton J A, Benson M D. Cell. Mol. Life. Sci., 2001, 58: 1491.
[39]
Nelson R, Sawaya M R, Balbirnie M, Madsen A O, Riekel C, Grothe R, Eisenberg D. Nature, 2005, 435(7034): 773.
[40]
Sacchettini J C, Kelly J W. Nat. Rev. Drug Discov., 2002, 1(4): 267.
[41]
Jahn T R, Radford S E. Arch. Biochem. Biophys., 2008, 469(1): 100.
[42]
Arsequell G, Planas A. Curr. Med. Chem., 2012, 19: 2343.
[43]
Oza V B, Smith C, Raman P, Koepf E K, Lashuel H A, Petrassi H M, Chiang K P, Powers E T, Sachettinni J, Kelly J W. J. Med. Chem., 2002, 45(2): 321.
[44]
Adamski-Werner S L, Palaninathan S K, Sacchettini J C, Kelly J W. J. Med. Chem., 2004, 47: 355.
[45]
Klabunde T, Petrassi H M, Oza V B, Raman P, Kelly J W, Sacchettini J C. Nat. Struct. Biol., 2000, 7: 312.
[46]
Gales L, Macero-Ribeiro S, Arsequell G, Valencia G, Saraiva M J, Damas A M. Biochem. J., 2005, 388: 615.
[47]
Julius R L, Farha O K, Chiang J, Perry L L, Hawthorne M F. Proc. Natl. Acad. Sci. U. S. A., 2007, 104: 4808.
[48]
Hu Z H, Tang Y H, Wang H F, Zhang X, Lei M. Arch. Biochem. Biophys., 2008, 475(2): 140.
[49]
Yuan T H, Zhang X, Hu Z H, Wang F, Lei M. Biopolymers, 2012, 97(12): 998.
[50]
Yang M F, Lei M, Huo S H. Protein Sci., 2003, 12: 1222.
[51]
Correia B E. Protein Sci., 2006, 15: 28.
[52]
Yang M F, Lei M, Yordanov B, Huo S H. J. Phys. Chem. B, 2006, 110(12): 5829.
[53]
Steward R E, Armen R S, Daggett V. Pro. Eng. Des. Sel., 2008, 21: 187.
[54]
Wang H F, Tang Y H, Lei M. Arch. Biochem. Biophys., 2007, 466: 85.
[55]
He Y W, Niu C W, Li H, Wen X, Xi Z. Sci. China-Chem., 2013, 56(3): 286.
[56]
Mairal T, Nieto J, Pinto M, Almeida M R, Gales L, Ballesteros A, Barluenga J, Perez J J, Vazquez J T, Centeno N B, Saraiva M J, Damas A M, Planas A, Arsequell G, Valencia G. PLoS One, 2009, 4: e4124.
[57]
Sim?es C J, Mukherjee T, Brito R M, Jackson R M. J. Chem. Inf. Model., 2010, 50: 1806.