Fang G M, Li Y M, Shen F, Huang Y C, Li J B, Lin Y, Cui H C, Liu L. Angew. Chem. Int. Ed., 2011, 50: 7645.
[2]
Zheng J S, Tang S, Qi J Q, Wang Z P, Liu L. Nat. Protoc., 2013, 8: 2483.
[3]
Malins L R, Cergol K M, Payne R G. ChemBioChem, 2013, 14: 559.
[4]
Dumas A, Spicer C D, Gao Z H, Takehana T, Lin Y A, Yasukohchi T, Davis B G. Angew. Chem. Int. Ed., 2013, 52: 3916.
[5]
Fang G M, Cui H K, Zheng J S, Liu L. ChemBioChem, 2010, 11: 1061.
[6]
Zheng J S, Cui H K, Fang G M, Xi W X, Liu L. ChemBioChem, 2010, 11: 511.
[7]
Spokoyny A M, Zou Y K, Ling J J, Yu H T, Lin Y S, Pentelute B L. J. Am. Chem. Soc., 2013, 135: 5946.
[8]
McNaughton B R, Cronican J J, Thompson D B, Liu D R. Proc. Natl. Acad. Sci. U. S. A., 2009, 106: 6111.
[9]
Jenssen H, Aspmo S I. Methods Mol. Biol., 2008, 494: 177.
[10]
Schafmeister C E, Po J, Verdine G L. J. Am. Chem. Soc., 2000, 122, 5891.
[11]
Blackwell H E, Grubbs R H. Angew. Chem. Int. Ed., 1998, 37: 3281.
[12]
Baek S, Kutchukian P S, Verdine G L, Huber R, Holak T A, Lee K W, Popowicz G M. J. Am. Chem. Soc., 2012, 134: 103.
[13]
Phillips C, Roberts L R, Schade M, Bazin R, Bent A, Davies N L, Moore R, Pannifer A D, Pickford A R, Prior S H, Read C M, Scott A, Brown D G, Xu B, Irving S L. J. Am. Chem. Soc., 2011, 133: 9696.
[14]
Bernal F, Tyler A F, Korsmeyer S J, Walensky L D, Verdine G L. J. Am. Chem. Soc., 2007, 129: 2456.
[15]
Moellering R E, Cornejo M, Davis T N, Bianco C D, Aster J C, Blacklow S C, Kung A L, Gilliland D G, Verdine G L, Bradner J E. Nature, 2009, 462: 182.
[16]
Zhang H, Zhao Q, Bhattacharya S, Waheed A A, Tong X, Hong A, Heck S, Curreli F, Goger M, Cowburn D, Freed E O, Debnath A K. J. Mol. Biol., 2008, 378: 565.
[17]
Bautista A D, Appelbaum J S, Craig C J, Michel J, Schepartz A. J. Am. Chem. Soc., 2010, 132: 2904.
[18]
Bird G H, Bernal F, Pitter K, Walensky L D. Methods Enzymol., 2008, 446: 369.
[19]
Gavathiotis E, Suzuki M, Davis M L, Pitter K, Bird G H, Katz S G, Tu H C, Kim H, Cheng E H, Tjandra N T, Walens L D. Nature, 2008, 455: 1076.
[20]
Pitter K, Bernal F, Labelle J, Walensky L D. Methods Enzymol., 2008, 446: 387.
[21]
Danial N N, Gramm C F, Scorrano L, Zhang C-Y, Krauss S, Ranger A M, Datta S R, Greenberg M E, Licklider L J, Lowell B B, Gygi S P, Korsmeyer S J. Nature, 2003, 424: 952.
[22]
Plas D R, Thompson C B. Trends Endocrin. Met., 2002, 13: 74.
[23]
Pinton P, Rizzuto R. Cell Death Differ., 2006, 13: 1409.
[24]
Sticht J, Humbert M, Findlow S, Bodem J, Muller B, Dietrich U, Werner J, Krausslich H G. Nat. Struct. Mol. Biol., 2005, 12: 671.
[25]
Cui H K, Qing J, Guo Y, Wang Y J, Cui L J, He T H, Zhang L Q, Liu L. Bioorg. Med. Chem., 2013, 21: 3547.
[26]
Thorstholm L, Craik D J. Drug Discov. Today Tech. 2012, 9: e13.
[27]
G?ransson U, Svang?rd E, Claeson P, Bohlin L. Curr. Protein Pept. Sci., 2004, 5: 317.
[28]
Tang Y Q, Yuan J, Osapay G, Osapay K, Tran D, Miller C J, Ouellette A J, Selsted M E. Science, 1999, 286: 498.
[29]
Dawson P E, Muir T W, Lewis L C, Kent S B H. Science, 1994, 266: 776.
[30]
Durek T, Torbeev V Y, Kent S B H. Proc. Natl. Acad. Sci. U. S. A., 2007, 104: 4846.
[31]
Torbeev V Y, Kent S B H. Angew. Chem. Int. Ed., 2007, 46: 1667.
[32]
McGinty R K, Kim J, Chatterjee C, Roeder R G, Muir T W. Nature, 2008, 453: 812.
[33]
Fang G M, Wang J X, Liu L. Angew. Chem. Int. Ed., 2012, 51: 10347.
[34]
Zheng J S, Chang H N, Wang F L, Liu L. J. Am. Chem. Soc., 2011, 133: 11080.
[35]
Zheng J S, Huang Y C, Tang S, Liu L. Acc. Chem. Res., 2013, 46: 2475.
[36]
Chen Y X, Koch S, Uhlenbrock K, Weise K, Das D, Gremer L, Brunsveld L, Wittinghofer A, Winter R, Triola G, Waldmann H. Angew. Chem. Int. Ed., 2010, 49: 6090.
[37]
Huang Y C, Li Y M, Chen Y, Pan M, Li Y T, Yu L, Guo Q X, Liu L. Angew. Chem. Int. Ed., 2013, 52: 4858.
[38]
Dawson P E, Kent S B H. Biochem., 2000, 69: 923.
[39]
Binschik J, Mootz H D. Angew. Chem. Int. Ed., 2013, 52: 4260.
[40]
Adams A L, Macmillan D. J. Pept. Sci., 2013, 19: 65.
[41]
Gordon W R, Bang D, Hoff W D, Kent S B H. Bioorg. Med. Chem., 2013, 21: 3436.
[42]
Li Y M, Yang M Y, Huang Y C, Li Y T, Chen P R, Liu L. ACS Chem. Biol., 2012, 7: 1015.
[43]
Cronican J J, Thompson D B, Beier K T, McNaughton B R, Cepko C L, Liu D R. ACS Chem. Biol., 2010, 5: 747.
[44]
Lawrence M S, Phillips K J, Liu D R. J. Am. Chem. Soc., 2007, 129: 10110.
[45]
Dastlik K A, Sundermerier U, Johns D M, Chen Y, Williams R M. Synlett, 2005, 4: 693.
[46]
Williams R M, Im M N. J. Am. Chem. Soc., 1991, 113: 9276.
[47]
Kim Y W, Grossmann T N, Verdine G L. Nat. Protoc., 2011, 6: 761.
[48]
Muppidi A, Li X L, Chen J D, Lin Q. Bioorg. Med. Chem. Lett., 2011, 21: 7412.
[49]
Greenfield N, Fasman G D. Biochem, 1969, 8: 4108.
[50]
Walensky L D, Kung A L, Escher I, Malia T J, Barbuto S, Wright R D, Wagner G, Verdine G L, Korsmeyer S J. Science, 2004, 305: 1466.
[51]
Verdine G L, Hilinski G J. Methods in Enzymology, 2012, 503: 3.
[52]
Stewart M L, Fire E, Keating A E, Walensky L D. Nat. Chem. Biol., 2010, 6: 595.
[53]
Walensky L D, Pitter K, Morash J, Oh K J, Barbuto S, Fisher J, Smith E, Verdine G L, Korsmeyer S J. Mol. Cell, 2006, 24: 199.
[54]
Bernal F, Wade M, Godes M, Davis T N, Whitehead D G, Kung A L, Wahl G M, Walensky L D. Cancer Cell, 2010, 18: 411.
[55]
Karbowski M, Norris K L, Cleland M M, Jeong S Y, Youle R J. Nature, 2006, 443: 658.
[56]
Sakalian M, McMurtrey C P, Deeg F J, Maloy C W, Li F, Wild C T, Salzwedel K. J. Virol., 2006, 80: 5715.
[57]
Bird G H, Madani N, Perry A F, Princiotto A M, Supko J G, He X Y, Gavathiotis E, Sodroski J G, Walensky L D. Proc. Natl. Acad. Sci. U. S. A., 2010, 107: 14093.
[58]
Cui H K, Zhao B, Li Y H, Guo Y, Hu H, Liu L, Chen Y G. Cell Res., 2013, 23: 581.
[59]
Cascales L, Craik D J. Org. Biomol. Chem., 2010, 8: 5035.
[60]
G?ransson U, Burman R, Gunasekera S, Str?mstedt A A, Rosengren K J. J. Biol. Chem., 2012, 287: 27001.
[61]
Zheng J S, Tang S, Guo Y, Chang H N, Liu L. ChemBioChem, 2012, 13: 542.
[62]
Cowper B, Craik D J, Macmillan D. ChemBioChem 2013, 14: 809.
[63]
Zheng J S, Chang H N, Shi J, Liu L. Sci. China Chem., 2012, 55: 64.
[64]
Daly N L, Rosengren K J, Craik D J. Curr. Protein Pept. Sci., 2004, 5: 297.
[65]
Cui H K, Guo Y, He Y, Wang F L, Chang H N, Wang Y J, Wu F M, Tian C L, Liu L. Angew. Chem. Int. Ed., 2013, 52: 9558.