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化学进展  2006 

99mTc放射性药物中的配位化学

, PP. 1615-1625

Keywords: 99mTc放射性药物,金属有机配合物,双功能螯合剂

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Abstract:

在99mTc间接标记放射性药物中双功能螯合剂起到重要的连接作用，其在很大程度上决定了放射性药物的理化性质。99mTc标记放射性药物中常用的双功能螯合剂大都含有N、S、P等杂原子，本文以与锝核配位杂原子的不同对双功能螯合剂进行分类，分别对NxS(4-x)型配体、“3＋1”混合配体、含膦配体以及以[99mTc(CO)3]+为配位中心的99mTc放射性药物逐一进行介绍。

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