[1] | [3 ] Hilgenbrink A R,Low P S. J. Pharm. Sci. ,2005,94: 2135—2146
|
[2] | [5 ] Ke C Y,Mathias C J,Green M A. Adv. Drug Deliv. Rev. ,2004,56: 1143—1160
|
[3] | [6 ] Gucalp R,Dutcher J,Wiernik P H. Semin. Nucl. Med. ,1997,27: 3—9
|
[4] | [7 ] Elnakat H,Ratnam M. Adv. Drug Deliv. Rev. ,2004,56:1067—1084
|
[5] | [8 ] Sudimack J,Lee R J. Adv. Drug Deliv. Rev. ,2000,41:147—162
|
[6] | Ross T L,Honer M,Schibli R. Bioconjugate Chem. ,2008,19:2462—2470
|
[7] | Leamon C P,Low P S. Biochem. J. ,1993,291: 855—860
|
[8] | Mathias C J,Wang S,Lee R J,et al. J. Nucl. Med. ,1996,37: 1003—1008
|
[9] | Wang S,Lee R J,Low P S,et al. Bioconjugate Chem. ,1996,7: 56—62
|
[10] | Mathias C J,Hubers D,Low P S,et al. Bioconjugate Chem. ,2002,11: 253—257
|
[11] | Mathias C J,Wang S,Water D J,et al. J. Nucl. Med. ,1998,39: 1579—1585
|
[12] | Ross T L, Honer M, Ametamey S M, et al. Bioconjugate Chem. ,2008,19: 2462—2470
|
[13] | Bettio A,Honer M,Muller C,et al. J. Nucl. Med. ,2006,47:1153—1160
|
[14] | Trump D P,Mathias C J,Yang Z F,et al. Nucl. Med. Biol. ,2002,29: 569—573
|
[15] | Müller C,Dumas C,Schibli R,et al. J. Organomet. Chem. ,2004,689: 4712—4721
|
[16] | Müller C,Hohn A,Schibli R,et al. Eur. J. Nucl. Med. Mol.Imaging,2006,33: 1007—1016
|
[17] | Müller C,Schubiger P A,Schibli R. Nucl. Med. Biol. ,2007,34: 595—601
|
[18] | Müller C, Schubiger P A, Schibli R. Bioconjugate Chem. ,2006,17: 797—806
|
[19] | Struthers H,Spingler B,Mindt T L,et al. Chem. Eur. J.2008,14: 6173—6183
|
[20] | Müller C,Forrer F,Schibli R,et al. J. Nucl. Med. ,2008,49: 310—317
|
[21] | Reddy J A,Xu L C,Parker N,et al. J. Nucl. Med. ,2004,45: 857—866
|
[22] | Sega E I,Low P S. Cancer Metastasis Rev. ,2008,27: 655—664
|
[23] | Okarvi S M,Jammaz I A. Cancer Biother. Radiopharm. ,2006,21: 49—61
|
[24] | 胡春林(Hu C L) ,崔海平( Cui H P) ,杜进( Du J) . 核化学与放射化学( Journal of Nuclear and Radiochemisty ) ,2007,29: 231—237
|
[25] | Wedeking P W, Wager R E, Arunachalam T, et al. US 6221334,2001
|
[26] | Guo W,Hinkle G H,Lee R J. J. Nucl. Med. ,1999,40:1563—1569
|
[27] | 刘丽琴( Liu L Q) ,王世真(Wang S Z) ,李方( Li F) 等. 中国医学科学院学报( Acta Acad. Med. Sin. ) ,2006,28: 786—789
|
[28] | 万丹晶(Wan D J) ,钟高仁( Zhong G R) ,朱建华( Zhu J H)等. 核技术(Nuclear Techiniques) ,2004,27: 293—296
|
[29] | Lui M,Xu W,Xu L J,et al. Bioconjugate chem. ,2005,16:1126—1132
|
[30] | [1 ] Sudimack J,Lee R J. Adv. Drug Deliv. Rev. ,2000,41147—162
|
[31] | [2 ] Ke C Y,Mathias C J,Green M A. Nucl. Med. Biol. ,2003,30: 811—817
|
[32] | [4 ] Leamon C P,Low P S. Drug Discovery Today,2001,6: 44—51
|
[33] | [9 ] Low P S,Antony A C. Adv. Drug Deliv. Rev. ,2004,56:1055—1058
|
[34] | Maziarz K M,Monaco H L,Ratnam M. J. Biol. Chem. ,1999,274: 11086—11901
|
[35] | Ke C Y,Mathias C J,Green M A. J. Am. Chem. Soc. ,2005,127: 7421—7426
|
[36] | Wang S,Lou J,Lantrip D A,et al. Bioconjugate Chem. ,1997,8: 673—679
|
[37] | Wang S,Luo J,Low P S. Bioconjugate Chem. ,1997,8: 673—679
|
[38] | Alberto R,Schibli R,Kaden T A. J. Am. Chem. Soc. ,1998,120: 7987—7988
|
[39] | Mindt T L,Struthers H,Schibli R,et al. J. Am. Chem. Soc. ,2006,128: 15096—15097
|
[40] | Mindt T L,Müller C,Schibli R,et al. Bioconjugate Chem. ,2008,19: 1689—1695
|
[41] | 刘伯里( Liu B L) ,贾红梅( Jia H M) . 锝药物化学及其应用( Technetium Radiopharmaceutical Chemistry and Its Applications) . 北京: 北京师范大学出版社( Beijing: Beijing Normal University Press) ,2006. 84—94
|
[42] | Leamon C P,Parker M A,Vlahov I R,et al. Bioconjugate Chem. ,2002,13: 1200—1210
|
[43] | Wedeking P W, Wager R E, Arunachalam T, et al. US 6093382,2000
|
[44] | Llgan S, Yang D J, Higuch T, et al. Cancer Biother.Radiopharm. ,1995,13: 427—435
|
[45] | Decristoforo C,Mather S J. Nucl. Med. Biol. ,1999,26:389—396
|
[46] | Mathias C J,Hubers D,Low P S,et al. Bioconjugate Chem. ,2000,11: 253—257
|
[47] | Leamon C P,You F,Krishna H. Pharm. Res. ,2009,26:1315—1323
|
[48] | Shen Y, Zhang Y, Sun Y, et al. J. Label. Comp.Radiopharm. ,2009,52( S1) : S101—S116
|
[49] | Müller C,Schibli R,Forrer F,et al. Nucl. Med. Biol. ,2007,34: 603—608
|
[50] | Müller C,Schibli R,Krenning E P,et al. J. Nucl. Med. ,2008,49: 623—629
|
[51] | Müller C,Mindt T L,Schibli R,et al. Eur. J. Nucl. Med.Mol. Imaging,2009,36: 938—946
|