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OALib Journal期刊
ISSN: 2333-9721
费用：99美元
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AmmoniumDihydrogenPhosphateCatalystforOne-PotSynthesisof3,4-Dihydropyrimidin-2(1H)-ones
DOI: 10.1016/S1872-2067(11)60355-0, PP. 659-665
Keywords: 3,4-dihydropyrimidin-2-(1H)-one,ammoniumdihydrogenphosphate,solventfree,condensation
Abstract:
？Aone-potthreecomponentBiginellicondensationofdifferentsubstitutedaromaticandaliphaticaldehydeswithethylacetoacetateandureatotherespective3,4-dihydropyrimidin-2-(1H)-onesundersolvent-freeconditionsthatissimple,effective,andenvironmentallyfriendlywasshown.Ammoniumdihydrogenphosphate(NH4H2PO4)wasusedasanon-toxic,inexpensive,andeasilyavailablecatalyst.Thefacilereactionconditionandsimpleisolationandpurificationproceduresofthismethodmakeitagoodoptionforthesynthesisofdihydropyrimidinones.
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