%0 Journal Article %T GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain %A Allan J. B. Watson %A Anne-Marie Michon %A Armelle Le Gall %A Chun-wa Chung %A Clare I. Hobbs %A Darren J. Mitchell %A David J. Fallon %A David Lugo %A Edward Hooper-Greenhill %A Emma J. Jones %A Emmanuel H. Demont %A Hawa Diallo %A Heather A. Barnett %A Isabelle Becher %A Laurie J. Gordon %A Mark J. Bird %A Paola Grandi %A Paul Bamborough %A Peter D. Craggs %A Rab K. Prinjha %A Robert J. Watson %A Robert P. Law %J Archive of "ACS Medicinal Chemistry Letters". %D 2016 %R 10.1021/acsmedchemlett.6b00092 %K BRPF1 %K BRPF2 %K BRD1 %K BRPF3 %K BET %K bromodomain %K epigenetics %K chemical probe %K inhibitor %U https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4904261/