%0 Journal Article %T Discovery of TAK-272: A Novel, Potent, and Orally Active Renin Inhibitor %A Craig A. Behnke %A Gyorgy Snell %A Hidekazu Tokuhara %A Keiji Kusumoto %A Mitsuyo Kondo %A Ray Kanagawa %A Yasuhiro Imaeda %A Yoshiyuki Fukase %A Yumiko Kajimoto %J Archive of "ACS Medicinal Chemistry Letters". %D 2016 %R 10.1021/acsmedchemlett.6b00251 %K Renin inhibitor %K TAK-272 %K benzimidazole %K hypertension %K SBDD %K dTg rat %U https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5066151/