%0 Journal Article %T Systematic Study of Effects of Structural Modifications on the Aqueous Solubility of Drug-like Molecules %A Brandon Q. Mercado %A Jos¨¦ A. Cisneros %A Michael J. Robertson %A William L. Jorgensen %J Archive of "ACS Medicinal Chemistry Letters". %D 2017 %R 10.1021/acsmedchemlett.6b00451 %K Aqueous solubility %K MIF inhibitors %K crystallography %U https://www.ncbi.nlm.nih.gov/pmc/articles/PMC5238483/