%0 Journal Article %T Discovery of Novel Tricyclic Heterocycles as Potent and Selective DPP-4 Inhibitors for the Treatment of Type 2 Diabetes %A Aileen Soriano %A Andrew Stamford %A Dmitri Pissarnitski %A Duane A. Burnett %A Giovanna Scapin %A Hong Mei %A Jinsong Hao %A Joyce Hwa %A Martin Domalski %A Mary Ann Powles %A Shiying Chen %A Terri M. Kelly %A Wen-Lian Wu %A Ying-Duo Gao %A Zhiqiang Zhao %A Zuliang Yao %J Archive of "ACS Medicinal Chemistry Letters". %D 2016 %R 10.1021/acsmedchemlett.6b00027 %K Diabetes %K dipeptidyl peptidase IV (DPP-4) %K inhibitor %K tricyclic heterocycles %K crystal structure %K OGTT %U https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4867478/