%0 Journal Article
%T Discovery of Benzotriazolo[4,3-d][1,4]diazepines as Orally Active Inhibitors of BET Bromodomains
%A Adrianne Neiss
%A Alexander M. Taylor
%A Alexandre C£¿t¨¦
%A Brian K. Albrecht
%A Christopher G. Nasveschuk
%A Eneida Pardo
%A Florence Poy
%A Hari Jayaram
%A James E. Audia
%A Jean-Christophe Harmange
%A Jennifer A. Mertz
%A Jeremy W. Setser
%A Jose M. Lora
%A Michael
C. Hewitt
%A Peter Sandy
%A Richard T. Cummings
%A Rishi G. Vaswani
%A Robert
J. Sims
%A III
%A Shivangi Joshi
%A Steve Bellon
%A Victor S. Gehling
%A Yong Tang
%A Yves Leblanc
%J Archive of "ACS Medicinal Chemistry Letters".
%D 2016
%R 10.1021/ml500411h
%K Bromodomain
%K IL-6 inhibition
%K BRD4
%K BET
%U https://www.ncbi.nlm.nih.gov/pmc/articles/PMC4753545/