%0 Journal Article
%T Synthesis of 2-(6-Acetamidobenzothiazolethio)acetic Acid Esters as Photosynthesis Inhibitors
%A Eva Sidoova
%A Katarina Kralova
%A Dusan Loos
%J Molecules
%D 1998
%I MDPI AG
%R 10.3390/30400135
%X The synthesis and photosynthesis-inhibiting activity of 13 new 2-(6-acetamidobenzothiazolethio)acetic acid esters are reported. The new compounds were prepared by acetylation of 2-(alkoxycarbonylmethylthio)-6-aminobenzothiazoles with acetic anhydride. The structure of the compounds was verified by 1H NMR spectra. The compounds inhibit photosynthetic electron transfer in spinach chloroplasts. The structure - activity relation was studied. Lipophilicity was found to influence substantially photosynthetic electron transfer.
%K Electron transfer inhibition
%K QSAR
%K lipophilicity
%U http://www.mdpi.com/1420-3049/3/4/135